Custom Peptides
Cayman Chemical EmodIn 8-glucosIde 10mg
An anthraquinone glycoside; inhibits the activities of rat lens aldose reductase and human DNA topoisomerase II (IC50s = 14.4 and 66 μM, respectively, in cell-free assays); promotes the proliferation and differentiation of mouse MC3T3-E1 osteoblastic cells at 1 ng/ml; decreases infarct size in a rat model of focal cerebral ischemia and reperfusion injury at 5 mg/kg
Cayman Chemical ErythrodIol 10mg
A triterpene with diverse biological activities; induces relaxation of isolated rat aortic rings precontracted with phenylephrine (EC50 = 3.38 µM); inhibits the growth of HT-29 adenocarcinoma cells (EC50 = 48.8 µM); induces production of ROS and apoptosis in MCF-7 cells at 100 µM; topical administration reduces TPA-induced EAr edema and MPO activity in mice at 0.5 mg/ear
Cayman Chemical PIbrentasvIr 10mg
An HCV NS5A inhibitor; inhibits HCV replication in stable replicon cell lines containing NS5A from genotypes 1-6 (EC50s = 1.4-4.3 pM); acts synergistically with glecaprevir to inhibit HCV genotype 1b-Con1 replication in replicon cells
Cayman Chemical ngenol-3-ngelate 10mg
A hydrophobic diterpene ester that rapidly induces cell death in proliferating keratinocytes through plasma membrane and mitochondrial disruption; causes inflammation due, at least in part, to activation of PKC, leading to antibody-dependent cellular cytotoxicity
Cayman Chemical ElvItegravIr 10mg
A quinolone antibiotic that inhibits HIV-1 integrase (IC50 = 7.2 nM); has antiviral activity against laboratory strains and clinical isolates of HIV-1 in MAGI cells (EC50s = 0.1-1.26 nM) and HIV-2 in PBMCs (EC50s = 0.3-0.9)
Cayman Chemical 3FluoromethamphetamInhydr 10mg
An isomer of 4-FMA characterized by having fluorine at the 3 position of the phenyl group; intended for forensic and research applications
Cayman Chemical SynthetIc HIspolon 10mg
A phenol with diverse biological activities; scavenges superoxide and hydroxyl radicals in cell-free assays, as well as reduces LPS-induced production of ROS in RAW 264.7 cells at 5 and 10 µM; inhibits cell proliferation and induces apoptosis in C6 rat glioma and DBTRG-05MG human glioblastoma cells from 60-80 µM; reduces acetic acid-induced writhing in mice at 20 mg/kg
Cayman Chemical 2-AIhydrochlorIde 10mg
An aminoindane that serves as the starting point for the synthesis of psychoactive compounds, such as 5,6-methylenedioxy-2-aminoindane; has modest analgesic and stimulatory properties; intended for forensic applications
Cayman Chemical N NDImethylcathInonhydroc 10mg
A psychotropic compound of the phenethylamine and cathinone classes; slightly less potent than methcathinone and essentially equipotent with cathinone, in behavioral studies involving rats; intended for forensic purposes
Cayman Chemical 1 2DIlInoleoyl3aLInolenoy 10mg
A triacylglycerol; has been found in corn and soybean oils
Cayman Chemical Lnsoprazole sulfon NoxIde 10mg
A potential impurity found in commercial preparations of lansoprazole
Cayman Chemical FlavoxatehydrochlorIde 10mg
An inhibitor of L-type calcium channels and an antimuscarinic agent; induces relaxation of potassium-precontracted isolated human urinary bladder detrusor muscle (IC50 = 2 µM) and reduces carbachol- or calcium-induced contractions in isolated rat detrusor strips; inhibits reflex micturition in decerebrated cats when microinjected into the oral pontine reticular nucleus at 0.68 UG/animal
Cayman Chemical CGS 21680hydrochlorIde 10mg
A potent, selective agonist of the adenosine A2A receptor (Ki = 11-46 nM); less effective at adenosine A1 and A3 receptors (Kis = 0.5-3.1 and 0.6-1 µM, respectively) and is without effect at adenosine A2B (Ki > 10 µM)
Cayman Chemical 71 1HTetrazolylACTAmIdo 10mg
A potential impurity in commercial preparations of cefazolin